| 产品编号 | CFN60026 | |
| CAS编号 | 252917-06-9 | |
| 分子式 = 分子量 | C22H18Cl2N8 = 465.34 | |
| 产品纯度 | >=98% | |
| 物理属性 | Powder | |
| 化合物类型 | Alkaloids | |
| 植物来源 | ||
| ChemFaces的产品在影响因子大于5的优秀和顶级科学期刊中被引用 | ||
| 产品名称 | 产品编号 | CAS编号 | 包装 | QQ客服 |
| CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 1mg | QQ客服:215959384 |
| CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 5mg | QQ客服:215959384 |
| CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 10mg | QQ客服:215959384 |
| CHIR-99021 (CT99021) | CFN60026 | 252917-06-9 | 20mg | QQ客服:215959384 |
Cell. 2018 Jan 11;172(1-2):249-261.e12. doi: 10.1016/j.cell.2017.12.019.IF=36.216(2019)
Cell Metab. 2020 Mar 3;31(3):534-548.e5. doi: 10.1016/j.cmet.2020.01.002.IF=22.415(2019)
Mol Cell. 2017 Nov 16;68(4):673-685.e6. doi: 10.1016/j.molcel.2017.10.022.IF=14.548(2019)| Description: | CHIR-99021 (CT99021) is a GSK-3α and GSK-3β inhibitor with IC50 of 10 nM and 6.7 nM, respectively. CHIR99201 does not exhibit cross-reactivity against cyclin-dependent kinases (CDKs) and shows a 350-fold selectivity toward GSK-3β compared to CDKs. CHIR99021 functions as a Wnt/β-catenin activator and induces autophagy. |
| Targets: | GSK-3α/GSK-3β | CDK | Autophagy |
| 1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
| 1 mM | 2.149 mL | 10.7448 mL | 21.4897 mL | 42.9793 mL | 53.7242 mL |
| 5 mM | 0.4298 mL | 2.149 mL | 4.2979 mL | 8.5959 mL | 10.7448 mL |
| 10 mM | 0.2149 mL | 1.0745 mL | 2.149 mL | 4.2979 mL | 5.3724 mL |
| 50 mM | 0.043 mL | 0.2149 mL | 0.4298 mL | 0.8596 mL | 1.0745 mL |
| 100 mM | 0.0215 mL | 0.1074 mL | 0.2149 mL | 0.4298 mL | 0.5372 mL |
| 产品名称 | 产品编号 | CAS编号 | 分子式 = 分子量 | 位单 | 联系QQ |
| 3-(羟甲基)-3-硝基-1-(4-辛基苯基)-1,4-丁二醇; 3-(Hydroxymethyl)-3-nitro-1-(4-octylphenyl)-1,4-butanediol | CFN90100 | 899822-99-2 | C19H31NO5 = 353.45 | 5mg | QQ客服:2159513211 |
| 邻羟基苯乙酮; Ortho-Hydroxyacetophenone | CFN93191 | 118-93-4 | C8H8O2 = 136.2 | 20mg | QQ客服:1413575084 |
| RAF265 (CHIR-265); RAF265 (CHIR-265) | CFN60398 | 927880-90-8 | C24H16F6N6O = 518.41 | 5mg | QQ客服:2159513211 |
| LY294002; LY294002 | CFN60015 | 154447-36-6 | C19H17NO3 = 307.34 | 5mg | QQ客服:2056216494 |